A simple, facile and highly efficient one-pot approach has been unfolded for the syntheses of β-carboline tethered imidazole derivatives. Importantly, the β-carboline tethered imidazole derivatives displayed excellent photoph...
Artikel
Synthesis of Thienyl Polycyclic Fused Indoles Based on the Indium Catalyzed Prins/Friedel‐Crafts Tandem Reaction
Von Wiley-VCH zur Verfügung gestellt
An indium catalyzed Prins/Friedel-Crafts tandem cyclization reaction has been developed, providing facile access to a variety of polycyclic indole frameworks with high diastereoselectivity and good functional group tolerance.
Abstract
An indium catalyzed Prins/Friedel-Crafts tandem cyclization reaction has been developed. This reaction provides an efficient and practical method to construct a variety of polycyclic indole frameworks with high diastereoselectivity and good functional group tolerance (30 examples, up to 98% yield with >95 : 5 dr). The resulting products are easily accessible for further chemical transformations.
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